通过电介导的C-H转化区域选择性合成2，3'-二吲哚衍生物
Regioselective synthesis of toward 2,3'-biindoles via Electro-induced direct C-H transformations
目前关于电化学活化C-H键构建化合物是有机合成中的研究热点。本文首次报道了一种电化学方法，诱导N保护的吲哚衍生物的自身偶联，区域选择性合成了具有潜在生物活性的2,3'-二吲哚衍生物。这种电化学合成反应具有反应条件温和、操作简单、反应进程能够精确控制等优点。
t present, researchers have a strong interest in the organic synthesis constructed via Electro-induced C-H transformations. In this paper，we first report an electrochemical method that induces the homo-coupling of N-protected indole derivatives and regioselectively synthesizes 2,3'- biindole derivatives with potential biological activity. The electrochemical synthesis reaction has the advantages of mild reaction conditions, simple operation, and precise control of the reaction process.
秦波、李惠炼
电化学工业有机化学工业
电化学合成-H活化偶联反应2，3'-二吲哚衍生物
Electrochemical synthesisC-H activationcoupling reaction23'-biindoles
秦波,李惠炼.通过电介导的C-H转化区域选择性合成2，3'-二吲哚衍生物[EB/OL].(2019-03-19)[2025-08-11].http://www.paper.edu.cn/releasepaper/content/201903-250.点此复制
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